In the article, we will consider how to drink Afobazole in tablets.
Many people experience stress, anxiety, and excitement at times. And if methods such as a change of scenery and relaxation do not help, then you have to use medicines.
In modern pharmacology, there are many drugs to relieve stress and anxiety. They, as a rule, are among the tranquilizers. Their overwhelming amount depresses the nervous system and suppresses negative emotions. Their action is very powerful, and therefore they have long been used in the medical practice of psychotherapists and neuropathologists. Unfortunately, the disadvantage of these drugs is a large number of side effects.
However, in recent years, many “soft” tranquilizers have been developed, devoid of the above disadvantages. Such tranquilizers are often called "daytime". Afobazole, developed by Russian pharmacologists not so long ago, but already gained wide popularity, also belongs to them.
Structure
How to drink Afobazole in tablets is interesting to many.
The drug has a complex composition, as it includes the active substance and several auxiliary substances. The active ingredient is 5-ethoxy-2- [2- (morpholino) ethylthio] benzimidazole dihydrochloride, which is a derivative of anxiolytic - 2-mercaptobenzimidazole, which has a selective effect. The tablets also contain other substances: magnesium stearate; povidone; milk sugar; microcrystalline cellulose; potato starch.
Mechanism of action and features
How many Afobazole tablets to drink per day? We will talk about this below.
Patients familiar with the influence of tranquilizers of the old generation are well aware of the effect of the use of benzodiazepines - indifference to everything, detachment, lethargy. This is not a complete list of unpleasant symptoms of such drugs. Their most unpleasant feature is the formation of drug dependence in many patients, which, in particular, is reflected in the “withdrawal syndrome”, in which their condition worsens after treatment is stopped. Very often they become so attached to the tranquilizer that they can not imagine their life without it.
Afobazole has no such drawbacks. The drug does not affect the state of the nervous system, does not reduce the speed of the reaction, does not dull emotions, does not reduce the efficiency of the mind. Most importantly, he has no withdrawal syndrome. Thus, the patient can interrupt the treatment course at any time, and at the same time he will not have a craving for medicine. Upon completion of therapy, a gradual reduction in dosage is also not required to get rid of addiction. But, of course, it is important to know how many Afobazole tablets to drink per day for the best result.
The medication is also devoid of a large number of undesirable effects, practically has no contraindications. The drug is largely due to this can be dispensed without a prescription.
Its active ingredient does not affect benzodiazepine receptors, but it acts on the sigma-1 receptors in the brain. Receptors are responsible for sensory, emotions, fine motor skills and memory functioning. The drug has a slight anti-anxiety effect, activating along with this the nervous processes. Afobazole also enhances the bioenergetic potential of brain cells and has a neuroprotective effect, protecting neurons. A very weak sedative effect, it is felt only if the dosage exceeds the usual 40-50 times.
After administration, the drug is absorbed from the gastrointestinal tract with high speed. The average retention time in the patient's body is 1.6 hours. Differs in low toxicity. It is mainly metabolized in the liver.
How many Afobazole tablets can be drunk per day are indicated in the instructions.
Effects of use
The positive effect of the drug is expressed in the form of the following improvements:
- sleep improvement (if there is no daytime drowsiness);
- disappearance of preoccupation, fear, anxiety;
- elimination of psychological discomfort and nervous tension;
- decrease in disorders of the autonomic system (dizziness, sweating, dry mouth);
- improved attention and memory.
The greatest impact will be on patients with an asthenic type of nervous system. Such people are distinguished by the following features: vulnerability, suspiciousness, emotional lability, predisposition to stressful reactions, self-doubt.
Indications
The drug "Afobazole" is used in the presence of the following indications:
- adaptation violations;
- general anxiety disorder;
- cardiopsychoneurosis;
- insomnia;
- withdrawal syndrome during nicotine addiction therapy;
- neurasthenia;
- tension syndrome before menstruation;
- withdrawal syndrome with alcoholism.
The tool is also often used to stop anxiety, depression and fear caused by somatic diseases:
- arrhythmia;
- oncological pathologies;
- asthma;
- coronary heart disease;
- hypertension.
Practice shows that the greatest effect from the use of the drug is noted when relieving anxiety and depression in patients who suffer from diseases of the heart and blood vessels.
So, how to drink "Afobazole" in tablets?
Instructions for use, dosage
The drug should be taken three times a day after meals. The optimal dose is 30 mg, that is, three 10 mg tablets. In some cases, the dosage can be increased to 60 mg. But it’s best to tell how to drink Afobazole in tablets, only the attending physician can.
According to the instructions that come with the drug, the recommended dosage for suppressing a hangover syndrome is five to ten milligrams twice a day. The treatment course is determined by the prescription of a specialist, but usually lasts from two to four weeks. The course can be extended if necessary. But before resuming treatment, it is advisable to take a break for three to four weeks.
"Afobazole" can you drink 2 tablets? For some patients, two pills per day are enough; for others, a dosage of two tablets three times a day is suitable.
It should be noted that the drug has a gradual effect. Its effect accumulates and begins to manifest itself only after some time after the start of use, often after a week. That is why, if the administration was started, but no improvement was observed in the first days, this does not mean that the drug is ineffective. It’s worth a little wait.
How much you can drink Afobazole tablets, we told. And is everyone allowed this drug?
Contraindications
The drug has the following contraindications:
- the use of the drug is not recommended during pregnancy;
- with breastfeeding and simultaneous use of the drug, it is advisable to switch to artificial mixtures for the baby;
- the drug is suitable only for adult patients; it cannot be used to treat minor patients.
This must be considered before taking.
Knowing how to drink Afobazole in tablets should be done in order to avoid side effects of the medicine.
Side effects
The medication has a small number of side effects. In rare cases, there are allergic reactions to substances in the composition, as well as a headache, usually passing by itself. The drug does not affect the reaction rate and attention, and therefore, during treatment, you can drive vehicles, manage complex mechanisms. In case of an overdose, there may be a sedation and drowsiness.
Interaction with other substances and medicines
One of the advantages of the drug is that it does not interact with ethanol. But you must understand that against the background of a therapeutic course, the use of alcoholic beverages is undesirable, since they neutralize the therapeutic effectiveness. Also minimized is the interaction with medications. When taken with Diazepam, its anxiolytic effect is enhanced. Increased anticonvulsant effect of "carbamazepine". Concomitant use with antidepressants is prohibited.
Analogs
Currently, there is the only structural analogue of the drug in tablet form - the drug "Fabomotizol". In the form of a concentrate for the manufacture of a solution for infusion, there is a structural analogue of Neurofazol.
Indirect analogues are other anxiolytics, especially those related to the number of “soft” tranquilizers, for example, Tenoten, Adaptol, or Grandaxin. It must be said that, in general, Afobazol has fewer side effects compared to other anxiolytics.
conclusions
Since the appearance of the drug, the spores around it do not stop. Reviews about the medicine are often directly opposite. So, many patients believe that it really helped them. However, some specialized specialists (psychiatrists, neuropathologists, neurologists and psychotherapists) do not share enthusiastic assessments. For example, it is said that the drug acts relatively weakly and helps only in mild cases of depressive states and anxiety disorders. In more serious forms of mental and nervous illness, the drug is ineffective. Many also note that the drug acts very selectively - approximately half of the patients did not feel any improvement. But no one denies the positive properties of the drug - the absence of dependence and the minimum number of side effects.
That is why a reasonable question arises: do I need to try Afobazole at all? In this case, you must understand that the drug is among the “soft” tranquilizers, which is unlikely to cope with significant disorders of the nervous system, for example, real depression, and not transient depressive states. "Afobazole" is a tool intended for patients with a healthy nervous system, experiencing difficult life periods and stresses - changing the environment, exams, somatic illness, family difficulties, etc. In such cases, the use of the drug is much more rational than the use of "heavy" drugs with a large number of side effects. In addition, despite the over-the-counter dispensing of the drug, it is highly recommended that they not be treated without medical advice.
We examined how to drink Afobazole in tablets.