What is the drug "Sustanon 250"? The instruction for this medication will be presented a little further. From the materials of this article you will learn about what indications the mentioned medicine has, whether it has contraindications and analogues, what will happen in case of an overdose and so on.
Release form, description, composition of the drug
Sustanon 250 contains such active components as testosterone propionate, testosterone isocapronate, testosterone phenylpropionate and testosterone decanoate. As for the additional ingredients, they use peanut butter, benzyl alcohol and nitrogen.
In what form is Sustanon 250 made? Reviews of experts indicate that this medication goes on sale in the form of an oil solution for intramuscular injection.
The drug has a yellow color (slightly colored) and is contained in white glass ampoules.
Pharmacological characteristics
What is the principle of action of the drug "Sustanon 250"? The instruction says that this medication is androgenic.
Testosterone is the main endogenous hormone that promotes the growth and development of the genitals of the stronger sex and their secondary sexual characteristics.
As you know, throughout the life of men, testosterone plays an indispensable role in the normal functioning of the testicles, prostate and seminal vesicles. This hormone supports sexual desire, erection and well-being.
Taking the Sustanon 250 medication with hypogonadism increases the concentration of androstenedione, testosterone, dihydrotestosterone and estradiol in the blood. In addition, the globulin levels that bind sex hormones, as well as follicle-stimulating and luteinizing hormones, decrease. Their level is restored to normal levels.
From the foregoing, we can safely conclude that during treatment with the drug in question, all signs of testosterone deficiency are significantly reduced. After therapy, patients may notice an increase in muscle mass and bone mineral density. That is why this medication is actively used in bodybuilding. By the way, in people with increased body weight, its decrease is observed.
Features of the medication
What features does Sustanon 250 have? Experts say that due to therapy, patients normalize their sexual functions. Also in their blood, the concentration of low and high density lipoproteins and triglycerides decreases. In addition, the concentration of hemoglobin and hematocrit in the human body increases.
Acceptance of this agent does not cause any changes in the prostatic specific antigen, as well as in the level of liver enzymes.
During treatment, some men may experience an enlargement of the prostate gland without any changes in its work.
If the drug is taken by hypogonadal patients with diabetes mellitus, then they often have a decrease in blood glucose levels, as well as an increase in sensitivity to insulin.
Reception of hormonal preparation by boys with growth retardation and puberty stimulates secondary sexual characteristics. If the medication was used by transgender women, then they have masculinization.
Pharmacokinetic properties of the oil solution
Sustanon 250 contains several testosterone esters. According to experts, they have different times of action. After entering the bloodstream, they give in to the process of hydrolysis.
When using a single dose of the drug in the blood of a man, the level of total testosterone begins to gradually increase. Its highest concentration is observed after 1-2 days. At the same time, testosterone levels return to lower limits after about 21 days.
The connection of testosterone with plasma proteins is very high (more than 97%). Before dihydrotestosterone and estriol, this hormone is metabolized naturally. The drug is excreted from the body with urine.
Indications for use
What are the uses of Sustanon 250 for? This drug is used during testosterone replacement treatment of the stronger sex, in which pathological conditions associated with secondary and primary hypogonadism are noted.
It should also be noted that the medicine can be used to treat acquired or congenital hypogonadism.
Contraindications
The drug "Sustanon 250" is not prescribed in the following cases:
- in children under three years of age;
- with suspected breast or prostate cancer, as well as with an already established diagnosis;
- with a high sensitivity of the patient to any of the components of the drug.
This drug is prescribed with extreme caution in the prepubertal period in boys (it is necessary to avoid closing of the pineal glands and premature puberty).
In addition, with extreme caution, Sustanon 250 is used for chronic heart, liver or kidney failure, diabetes mellitus, apnea, prostate hypertrophy with urinary retention, chronic lung pathologies and obesity.
How to take "Sustanon 250"?
According to the instructions, such a solution should be administered deeply, intramuscularly. The dosage of Sustanon 250 should be determined only by an experienced physician. As a rule, it depends on the patient's response to treatment.
Most often, experts prescribe the next dose - one milliliter once every three weeks.
In bodybuilding, this drug can be used both solo and in combination with other medicines. For example, the Sustanon course is often practiced along with Deca Methane, Methane Sustanon and others.
Overdose cases
Now you know how to stab Sustanon 250. When using high doses of an intramuscular solution, the patient exhibits priapism. In this case, you must stop using the medicine until this symptom completely disappears. Resume administration of the drug is required already in smaller doses.
Side effects
What undesirable effects occur when using the drug "Sustanon 250"? A side effect can occur only if the medication was used in high doses. These reactions include the following:
- polycythemia;
- the occurrence of neoplasms (malignant, benign or uncertain);
- increase in blood pressure;
- prostate cancer or worsening of patients with prostate cancer;
- nausea;
- fluid retention in the body and the appearance of edema;
- nervous irritability, depressive states, changes in mood;
- decreased or increased sexual desire;
- myalgia;
- violation of the liver;
- itching, rash on the skin;
- oligospermia, gynecomastia, sperm reduction, prostate hypertrophy, priapism;
- hypercalcemia.
It should also be noted that after an intramuscular injection, the patient may manifest undesirable local reactions (itching, pain, redness).
Special recommendations for the use of the drug
Patients who have been prescribed the drug "Sustanon-250" should be regularly observed by a specialist. Doctors are required to monitor by means of a digital examination in order to exclude the development of benign prostatic hyperplasia.
In people with diseases of the kidneys, heart, and liver, complications in the form of acute heart failure and edema can be noted while taking the medicine.
If the medication was prescribed for elderly patients, it must be borne in mind that treatment with Sustanon-250 can increase the risk of developing prostate cancer and prostate hypertrophy.
Similar means and price of Sustanon-250
The analogues of the Sustanon-250 drug are Omnadren 250, Sustaver from Vermoge, Testosterone Propionate solution and others.
The price of the medication in question is not very high. One package with a solution can be purchased for 250-300 rubles.
Patient reviews about the drug
Most often, reviews about the drug "Sustanon 250" leave athletes. The popularity of this medication among athletes is growing every year more and more. They note its effective and quick action. The use of intramuscular injections in the recommended dosage leads to increased male strength and active muscle building.
According to the reviews of athletes, in order to achieve greater effectiveness in bodybuilding, Sustanon 250 must be combined with such means as Boldenon, Winstrol and others.
Despite the popularity of the drug among athletes, experienced specialists highly recommend not practicing the intake of androgens in order to build muscle. This is due to the fact that this drug has a large number of serious side effects (up to the development of malignant neoplasms).
It should also be noted that there are quite a lot of positive reviews about this medicine, which are left by patients who use it to improve their health with testosterone replacement treatment.