Hemorrhoids are a common ailment among both men and women of different ages. This problem is considered quite intimate, therefore, not every person visits a medical specialist when a disease occurs.
To eliminate pain, creams and ointments with an analgesic effect should be used. One of the most effective and safest is Papaverine. In most cases, ointment is used for external hemorrhoids.
In rare situations, hemorrhoids lead to complications that can occur if the inflamed nodes are not treated for a long period. Therefore, timely treatment of the disease is important. To do this, you need to select only highly effective and safe medicines.
Most medical professionals approve and prescribe papaverine-based drugs to their patients. As you know, it helps to effectively cope with unpleasant symptoms and pain. What is part of papaverine ointment?
Description
The active substance is papaverine hydrochloride. It is an opium alkaloid from the group of myotropic antispasmodics.
Auxiliary components are also included in the ointment "Papaverine":
- lanolin;
- sunflower oil;
- water.
With the help of this composition, the medication has a soft structure.
Pharmacological properties
Since papaverine is present in the preparation, the agent has analgesic and antispasmodic effects. Its effect is aimed at eliminating smooth muscle pain and spasm. Additional substances help eliminate constipation, as well as soothe and soften the epidermis.
Papaverine ointment relaxes smooth muscles. Sunflower oil exhibits a laxative effect, thereby preventing intestinal obstruction. Lanolin helps soften the skin. The drug forms a protective shell, preventing repeated irritation.
After use, the medicine is immediately absorbed by the walls of the rectum. Penetrates into the blood and binds to plasma proteins. It begins to act after 15-20 minutes. The positive effect lasts about 2 hours.
The lanolin included in the structure softens the epidermis and also prevents irritation. Sunflower oil has a laxative effect, thereby helping to prevent constipation. Active ingredients to a small extent pass through the liver. They are eliminated from the body by the kidneys together with urine in the form of metabolic products.
Indications for use of papaverine ointment
The annotation states that the medicine is prescribed for the following ailments:
- Smooth muscle stenosis in the intestinal canal.
- Spastic constipation (insufficient, delayed or difficult bowel movements, which is caused by spasms of the smooth muscles of the intestine).
- Pain in the veins.
- Spasms in the urethra.
- Stenosis in the anorectal region.
- Dermatitis (an inflammatory lesion of the skin resulting from exposure to damaging factors of a chemical, physical or biological nature).
Papaverine-based drugs are absolutely non-toxic, and they act instantly.
With hemorrhoids
With varicose veins of the venous plexus of the rectum, papaverine ointment is included in the structure of complex treatment. The medication has analgesic, as well as antispasmodic and sedative effects.
Ointment is often used to eliminate enlarged hemorrhoids. The drug is easy to use, while it dries quickly. A positive effect occurs 15-20 minutes after application. A person feels that pain, as well as itching and burning, begin to disappear.
An ointment with papaverine is prescribed for spastic constipation. The medicine is used for stenosis in the urethra. According to the instructions for use, papaverine ointment is indicated for application with a painful feeling in the veins.
With chronic varicose veins of the venous plexus of the rectum, the ointment acts as a sedative. There are substances in the structure that help prevent constipation of spastic origin.
In addition, with hemorrhoids, a lanolin ointment is used. It can be used on veins, which helps to dilate blood vessels and improve blood flow. The drug is often used to eliminate pain in hemorrhoids. But in such situations, rectal suppositories are recommended for use, which fall deep into the rectum and dissolve there.
But the medication can be used with an increase in external hemorrhoidal nodes. After applying "Papaverine" pain and discomfort are eliminated. The blood flow in the veins resumes, with the help of which the nodes are reduced in size.
Before using the medication, wash the sphincter area with soap and water. Ointment can be used with an increase in external hemorrhoidal nodes. After applying the medicine to the affected area, the patient should rest for 10-15 minutes.
How to apply ointment
Before using the drug, it is necessary to wash the area of the anus with water and soap. Then gently pat dry with a soft towel or paper towel. The patient takes a horizontal position, applies ointment to the affected area and rests for 10-15 minutes.
Repeat manipulations should be up to 2-3 times a day. The next application is possible 4 hours after use. The duration of the treatment course is from one to two weeks, depending on the course of the disease.
Contraindications
The drug is not allowed to be used by all patients. There are several limitations in the form:
- Severe liver failure.
- Increased susceptibility to the components of the ointment.
- Angle-closure glaucoma (an ophthalmic disease in which the level of intraocular pressure rises).
- Shock state.
- Renal failure.
- Traumatic brain injury.
- Thyroid disease.
- Cramping of cerebral vessels.
With extreme caution, the medicine should be used in cases of impaired cardiac conduction and kidney damage.
Angle-closure glaucoma is a limitation to the use of ointment. In addition, the drug is contraindicated in traumatic brain injury. Papaverine ointment is not recommended for cerebral stenosis.
Side effects of ointment "Papaverine"
During therapy, negative signs may occur, which manifest themselves in the form of:
- Drowsiness.
- Dizziness.
- Nausea and abdominal pain.
- Lowering blood pressure.
- Hyperhidrosis (increased sweating).
- Atonic constipation (the most common type of bowel disorder, occurs in people with a sedentary lifestyle).
Lanolin ointment can also provoke side effects: allergic reactions, which are accompanied by skin rashes, itching, burning, and hyperemia.
Application features
Ointment is allowed for use by women during pregnancy. But the concentration and duration of therapy is selected by a medical specialist, since the active component (papaverine) penetrates to a small degree into the blood and passes through the placenta.
The drug is allowed to be used with breastfeeding. During treatment, lactation can not be stopped. It is known that papaverine ointment is contraindicated in treating children under 3 years of age. In pediatrics is used very rarely.
Interaction with other medicines
If papaverine ointment is used simultaneously with Methyldopa and Levodopa, then a decrease in therapeutic effect is observed. Barbiturate increases the effect of the active substances of the ointment. Sedatives cause a hypotensive effect.
Generics
Papaverine medicines are very popular among patients. This is due to the increased safety and cost of the drug. But medications in the form of ointments, except for "Papaverine", do not exist. As substitutes, you can buy pills or candles.
Keep the ointment in its original packaging in a cool and dark place away from children. Shelf life is 2 years. The drug is dispensed without a prescription from a specialist.
Opinions
Reviews about the medicine can be found in different forums, since a wide range of pharmacological effects of papaverine (active component) helps to evaluate its effectiveness for a large audience of people with various diseases. Papaverine ointment for dermatitis, as well as hemorrhoids, is actively used.
For example, the medicine got positive responses from proctologists and their patients, since the drug is used as a symptomatic conservative therapy for hemorrhoids, one of the most pressing problems of our time. The use of a medicinal product in the form of an ointment helps to ease bowel movements, partially eliminate pain, as well as the problem of bleeding from dilated hemorrhoids.
On the other hand, one can observe positive responses about the liniment during pregnancy, since the antispasmodic and relaxing effects of the active ingredient component help to effectively eliminate uterine hypertonicity, which eliminates the threat of premature birth. "Papaverine" allows you to alleviate the cramping pain that accompanies the last weeks and days of bearing the baby. In addition, the pharmaceutical agent is used for prevention in hospitals.